Detalles de la búsqueda
1.
Design, synthesis, and biological screening of a series of 4'-fluoro-benzotriazole-acrylonitrile derivatives as microtubule-destabilising agents (MDAs).
J Enzyme Inhib Med Chem;
37(1): 2223-2240, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35979600
2.
Quinoxaline-based efflux pump inhibitors restore drug susceptibility in drug-resistant nontuberculous mycobacteria.
Arch Pharm (Weinheim);
355(8): e2100492, 2022 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-35532283
3.
Covalent Reversible Inhibitors of Cysteine Proteases Containing the Nitrile Warhead: Recent Advancement in the Field of Viral and Parasitic Diseases.
Molecules;
27(8)2022 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-35458759
4.
Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity.
Molecules;
27(2)2022 Jan 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-35056779
5.
Biological Effects on µ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives.
Molecules;
26(18)2021 Sep 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-34576918
6.
Design, Synthesis, and Antiviral Activities of New Benzotriazole-Based Derivatives.
Pharmaceuticals (Basel);
16(3)2023 Mar 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-36986528
7.
A quinolin-8-ol sub-millimolar inhibitor of UGGT, the ER glycoprotein folding quality control checkpoint.
iScience;
26(10): 107919, 2023 Oct 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-37822503
8.
Antibiotics and Carbohydrate-Containing Drugs Targeting Bacterial Cell Envelopes: An Overview.
Pharmaceuticals (Basel);
15(8)2022 Jul 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-36015090
9.
Benzimidazole-2-Phenyl-Carboxamides as Dual-Target Inhibitors of BVDV Entry and Replication.
Viruses;
14(6)2022 06 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-35746771
10.
The green chemistry of chalcones: Valuable sources of privileged core structures for drug discovery.
Front Chem;
10: 988376, 2022.
Artículo
en Inglés
| MEDLINE | ID: mdl-36172001
11.
Crystal polymorphism in fragment-based lead discovery of ligands of the catalytic domain of UGGT, the glycoprotein folding quality control checkpoint.
Front Mol Biosci;
9: 960248, 2022.
Artículo
en Inglés
| MEDLINE | ID: mdl-36589243
12.
Human Enterovirus B: Selective Inhibition by Quinoxaline Derivatives and Bioinformatic RNA-Motif Identification as New Targets.
Pharmaceuticals (Basel);
15(2)2022 Jan 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-35215294
13.
A comprehensive assessment of a new series of 5',6'-difluorobenzotriazole-acrylonitrile derivatives as microtubule targeting agents (MTAs).
Eur J Med Chem;
222: 113590, 2021 Oct 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34139625
14.
Synthesis, Antitumor and Antiviral In Vitro Activities of New Benzotriazole-Dicarboxamide Derivatives.
Front Chem;
9: 660424, 2021.
Artículo
en Inglés
| MEDLINE | ID: mdl-34017818
15.
Inhibition of Enterovirus A71 by a Novel 2-Phenyl-Benzimidazole Derivative.
Viruses;
13(1)2021 Jan 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-33406781
16.
Clamping, bending, and twisting inter-domain motions in the misfold-recognizing portion of UDP-glucose: Glycoprotein glucosyltransferase.
Structure;
29(4): 357-370.e9, 2021 04 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33352114
17.
Preliminary Anti-Coxsackie Activity of Novel 1-[4-(5,6-dimethyl(H)- 1H(2H)-benzotriazol-1(2)-yl)phenyl]-3-alkyl(aryl)ureas.
Med Chem;
16(5): 677-688, 2020.
Artículo
en Inglés
| MEDLINE | ID: mdl-31878859
18.
5,6-Dichloro-2-phenyl-benzotriazoles: New Potent Inhibitors of Orthohantavirus.
Viruses;
12(1)2020 01 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-31968537
19.
Solid Lipid Nanoparticles as Formulative Strategy to Increase Oral Permeation of a Molecule Active in Multidrug-Resistant Tuberculosis Management.
Pharmaceutics;
12(12)2020 Nov 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-33255304
20.
Enhancement of antimicrobial activity of pump inhibitors associating drugs.
J Infect Dev Ctries;
13(2): 162-164, 2019 02 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-32036352